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Phase 1/2 study of acalabrutinib and the PI3K delta inhibitor ACP-319 in relapsed/refractory B-cell Non-Hodgkin lymphoma.

Title: Phase 1/2 study of acalabrutinib and the PI3K delta inhibitor ACP-319 in relapsed/refractory B-cell Non-Hodgkin lymphoma.
Authors: Barr PM; Wilmot Cancer Institute, University of Rochester Medical Center, Rochester, NY, USA.; Smith SD; University of Washington/Fred Hutchinson Cancer Research Center, Seattle, WA, USA.; Roschewski MJ; National Cancer Institute, Bethesda, MD, USA.; O'Brien SM; Chao Family Comprehensive Cancer Center, University of California-Irvine, Irvine, CA, USA.; Sharman JP; Willamette Valley Cancer Institute and Research Center, US Oncology Research, Eugene, OR, USA.; Melear JM; Texas Oncology, Austin, TX, USA.; Patel P; AstraZeneca, South San Francisco, CA, USA.; Calvo R; AstraZeneca, Gaithersburg, MD, USA.; Yang H; AstraZeneca, South San Francisco, CA, USA.; Spurgeon SE; Knight Cancer Institute, Oregon Health and Sciences University, Portland, OR, USA.
Source: Leukemia & lymphoma [Leuk Lymphoma] 2022 Jul; Vol. 63 (7), pp. 1728-1732. Date of Electronic Publication: 2022 Feb 24.
Publication Type: Clinical Trial, Phase I; Clinical Trial, Phase II; Letter; Research Support, Non-U.S. Gov't
Language: English
Journal Info: Publisher: Taylor & Francis Country of Publication: United States NLM ID: 9007422 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1029-2403 (Electronic) Linking ISSN: 10268022 NLM ISO Abbreviation: Leuk Lymphoma Subsets: MEDLINE
Imprint Name(s): Publication: [Philadelphia, PA] : Taylor & Francis; Original Publication: Chur ; New York : London, UK : Harwood Academic Publishers ; Distributed by STBS, 1989-
MeSH Terms: Lymphoma, B-Cell*/drug therapy ; Lymphoma, B-Cell*/pathology ; Phosphatidylinositol 3-Kinases*; Adenosine ; Benzamides ; Humans ; Pyrazines ; Quinolines
Substance Nomenclature: K72T3FS567 (Adenosine); 0 (Benzamides); EC 2.7.1.- (Phosphatidylinositol 3-Kinases); 0 (Pyrazines); 0 (Quinolines); 19DG7G1U5Q (N-(1-(7-fluoro-2-(pyridin-2-yl)quinolin-3-yl)ethyl)-9H-purin-6-amine); I42748ELQW (acalabrutinib)
Entry Date(s): Date Created: 20220224 Date Completed: 20220712 Latest Revision: 20260127
Update Code: 20260130
DOI: 10.1080/10428194.2022.2043301
PMID: 35200084
Database: MEDLINE

Clinical Trial, Phase I; Clinical Trial, Phase II; Letter; Research Support, Non-U.S. Gov't