| Title: |
Discovery and characterization of orally bioavailable 4-chloro-6-fluoroisophthalamides as covalent PPARG inverse-agonists |
| Authors: |
Orsi, Douglas L. a, 1; Ferrara, Steven J. a; Siegel, Stephan b; Friberg, Anders c; Bouché, Léa b; Pook, Elisabeth d; Lienau, Philip b; Bluck, Joseph P. b; Lemke, Christopher T. a; Akcay, Gizem e; Stellfeld, Timo c; Meyer, Hanna c; Pütter, Vera c; Holton, Simon J. c; Korr, Daniel c; Jerchel-Furau, Isabel e; Pantelidou, Constantia e; Strathdee, Craig A. f; Meyerson, Matthew f, g, h, i; Eis, Knut b; Goldstein, Jonathan T. f, ⁎ |
| Source: |
In Bioorganic & Medicinal Chemistry 15 January 2023 78 |
| Database: |
ScienceDirect |