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Synthesis and initial in vitro evaluation of PSMA-targeting ligands with a modified aromatic moiety at the lysine ε-nitrogen atom

Title: Synthesis and initial in vitro evaluation of PSMA-targeting ligands with a modified aromatic moiety at the lysine ε-nitrogen atom
Authors: Zyk, Nikolai Y.; Ber, Anton P.; Nimenko, Ekaterina A.; Shafikov, Radik R.; Evteev, Sergei A.; Petrov, Stanislav A.; Uspenskaya, Anastasia A.; Dashkova, Natalia S.; Ivanenkov, Yan A.; Skvortsov, Dmitry A.; Beloglazkina, Elena K.; Majouga, Alexander G.; Machulkin, Aleksei E.
Contributors: Russian Foundation for Basic Research; Ministry of Science and Higher Education of the Russian Federation; Council on grants of the President of the Russian Federation
Source: Bioorganic & Medicinal Chemistry Letters ; volume 71, page 128840 ; ISSN 0960-894X
Publisher Information: Elsevier BV
Publication Year: 2022
Collection: ScienceDirect (Elsevier - Open Access Articles via Crossref)
Document Type: article in journal/newspaper
Language: English
DOI: 10.1016/j.bmcl.2022.128840
Availability: http://dx.doi.org/10.1016/j.bmcl.2022.128840; https://api.elsevier.com/content/article/PII:S0960894X2200316X?httpAccept=text/xml; https://api.elsevier.com/content/article/PII:S0960894X2200316X?httpAccept=text/plain
Rights: https://www.elsevier.com/tdm/userlicense/1.0/ ; https://doi.org/10.15223/policy-017 ; https://doi.org/10.15223/policy-037 ; https://doi.org/10.15223/policy-012 ; https://doi.org/10.15223/policy-029 ; https://doi.org/10.15223/policy-004
Accession Number: edsbas.5CA88D6B
Database: BASE