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Atypical Genetic Basis of Pyrazinamide Resistance in Monoresistant Mycobacterium tuberculosis

Title: Atypical Genetic Basis of Pyrazinamide Resistance in Monoresistant Mycobacterium tuberculosis
Authors: Modlin, Samuel J.; Marbach, Tyler; Werngren, Jim; Mansjö, Mikael; Hoffner, Sven E.; Valafar, Faramarz
Contributors: HHS | NIH | National Institute of Allergy and Infectious Diseases
Source: Antimicrobial Agents and Chemotherapy ; volume 65, issue 6 ; ISSN 0066-4804 1098-6596
Publisher Information: American Society for Microbiology
Publication Year: 2021
Description: Pyrazinamide (PZA) is a widely used antitubercular chemotherapeutic. Typically, PZA resistance (PZA-R) emerges in Mycobacterium tuberculosis strains with existing resistance to isoniazid and rifampin (i.e., multidrug resistance [MDR]) and is conferred by loss-of-function pncA mutations that inhibit conversion to its active form, pyrazinoic acid (POA).
Document Type: article in journal/newspaper
Language: English
DOI: 10.1128/aac.01916-20
DOI: 10.1128/AAC.01916-20
Availability: https://doi.org/10.1128/aac.01916-20; https://journals.asm.org/doi/pdf/10.1128/AAC.01916-20
Rights: https://creativecommons.org/licenses/by/4.0/ ; https://journals.asm.org/non-commercial-tdm-license
Accession Number: edsbas.62FC69F2
Database: BASE