| Title: |
Synthesis, Characterization, and Preclinical Evaluation of a Small-Molecule Prostate-Specific Membrane Antigen-Targeted Monomethyl Auristatin E Conjugate |
| Authors: |
Machulkin, Aleksei E.; Uspenskaya, Anastasia A.; Zyk, Nikolay U.; Nimenko, Ekaterina A.; Ber, Anton P.; Petrov, Stanislav A.; Polshakov, Vladimir I.; Shafikov, Radik R.; Skvortsov, Dmitry A.; Plotnikova, Ekaterina A.; Pankratov, Andrei A.; Smirnova, Galina B.; Borisova, Yulia A.; Pokrovsky, Vadim S.; Kolmogorov, Vasilii S.; Vaneev, Alexander N.; Khudyakov, Alexander D.; Chepikova, Olga E.; Kovalev, Sergey; Zamyatnin Jr, Andrey A.; Erofeev, Alexander; Gorelkin, Petr; Beloglazkina, Elena K.; Zyk, Nikolay V.; Khazanova, Elena S.; Majouga, Alexander G. |
| Contributors: |
Russian Science Foundation; Russian Foundation for Basic Research; Ministry of Education and Science of the Russian Federation; Interdisciplinary Scientific and Educational School, Moscow University |
| Source: |
Journal of Medicinal Chemistry ; volume 64, issue 23, page 17123-17145 ; ISSN 0022-2623 1520-4804 |
| Publisher Information: |
American Chemical Society (ACS) |
| Publication Year: |
2021 |
| Document Type: |
article in journal/newspaper |
| Language: |
English |
| DOI: |
10.1021/acs.jmedchem.1c01157 |
| Availability: |
https://doi.org/10.1021/acs.jmedchem.1c01157; https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c01157 |
| Rights: |
https://doi.org/10.15223/policy-029 ; https://doi.org/10.15223/policy-037 ; https://doi.org/10.15223/policy-045 |
| Accession Number: |
edsbas.C22737E |
| Database: |
BASE |