| Title: |
Discovery of the First Potent Inhibitors of Mutant IDH1 That Lower Tumor 2-HG in Vivo |
| Authors: |
Popovici-Muller, Janeta; Saunders, Jeffrey O.; Salituro, Francesco G.; Travins, Jeremy M.; Yan, Shunqi; Zhao, Fang; Gross, Stefan; Dang, Lenny; Yen, Katharine E.; Yang, Hua; Straley, Kimberly S.; Jin, Shengfang; Kunii, Kaiko; Fantin, Valeria R.; Zhang, Shunan; Pan, Qiongqun; Shi, Derek; Biller, Scott A.; Su, Shinsan M. |
| Source: |
ACS Medicinal Chemistry Letters ; volume 3, issue 10, page 850-855 ; ISSN 1948-5875 1948-5875 |
| Publisher Information: |
American Chemical Society (ACS) |
| Publication Year: |
2012 |
| Document Type: |
article in journal/newspaper |
| Language: |
English |
| DOI: |
10.1021/ml300225h |
| Availability: |
https://doi.org/10.1021/ml300225h; https://pubs.acs.org/doi/pdf/10.1021/ml300225h |
| Accession Number: |
edsbas.D9ABAAC4 |
| Database: |
BASE |