| Title: |
Click. Screen. Degrade. A Miniaturized D2B Workflow for Rapid PROTAC Discovery |
| Authors: |
Mitrović, Marko; Greco, Francesco Aleksy; García, Yiliam Cruz; Lučić, Aleksandar; Hoffmann, Lasse; Chander, Rohit; Schönfeld, Julia; Liebisch, Nick; Sivashanmugam, Saran Aswathaman; Schwalm, Martin Peter; Egner, Markus; Lewandowski, Max; Merk, Daniel; Morasch, Viktoria; Wolf, Elmar; Müller, Susanne; Hanke, Thomas; Proschak, Ewgenij; Hiesinger, Kerstin; Knapp, Stefan |
| Contributors: |
Bayer; Deutschen Konsortium f??r Translationale Krebsforschung; Roche; Deutsche Forschungsgemeinschaft; Pfizer; Bristol Myers Squibb Foundation; Genome Canada; European Commission; Boehringer Ingelheim; Merck; Deutsche Krebshilfe; Takeda; Janssen |
| Source: |
Journal of Medicinal Chemistry ; volume 69, issue 3, page 2599-2624 ; ISSN 0022-2623 1520-4804 |
| Publisher Information: |
American Chemical Society (ACS) |
| Publication Year: |
2026 |
| Document Type: |
article in journal/newspaper |
| Language: |
English |
| DOI: |
10.1021/acs.jmedchem.5c02543 |
| Availability: |
https://doi.org/10.1021/acs.jmedchem.5c02543; https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5c02543 |
| Rights: |
https://creativecommons.org/licenses/by/4.0/ |
| Accession Number: |
edsbas.F3A7A507 |
| Database: |
BASE |